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" DE LEAN, A., STADEL, JM AND LEFKOWITZ, RJ: A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled beta-adrenergic receptor. "
Farmacología Humana - Página 17
por Jesús Flórez - 2003 - 1416 páginas
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Receptor Binding in Drug Research

A. O'brien - 1986 - 552 páginas
...chlorpromazine. J. Pharm. Pharmacol. 22:193-197. De Lean, A., Stadel, JM, and Lefkowtiz, RJ (1980). A ternary complex model explains the agonist-specific...cyclase-coupled beta-adrenergic receptor. J. Biol. Chem. 255:71087117. Enna, SJ, Bennett, JP, Jr., Burt, DR, Creese, I., and Snyder, SH (1976). Stereospecificity...
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Corticotropin-Releasing Factor

Errol B. De Souza, Charles B. Nemeroff - 1989 - 380 páginas
...primate brain, Proc. Natl. Acad. Sci. USA, 83, l92l, l986. 34. DeLean, A., Stadel, JM, and Lefkowitz, RJ, A ternary complex model explains the agonist-specific...binding properties of the adenylate cyclase-coupled p-adrenergic receptor, J. Biol. Chem., 255, 7l08, l980. 35. ( 'rawIcy, JN, Olschowka, JA, Diz, DI,...
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Thermodynamics of Membrane Receptors and Channels

Meyer B. Jackson - 1992 - 454 páginas
...binding of I25Iglucagon, J Biol Chem., 246, 1872, 1971. 18. De Lean, A., Stadel, .IM, and Lefkowitz, RJ, A ternary complex model explains the agonist-specific...binding properties of the adenylate cyclase-coupled p-adrenergic receptor, J Biol Chem., 255, 7108, 1980. 19. Schramm, M. and Selinger, Z., Message transmission:...
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Molecular Biology of Membranes

H.R. Petty - 1993 - 432 páginas
...the hamster a,-adrenergic receptor. Proc. Natl. Acad. Sci. USA 85:7159-7163. DeLean, A., et al. 1980. A ternary complex model explains the agonist-specific...binding properties of the adenylate cyclase-coupled p-adrenergic receptor. J. Biol. Chem. 255:7108-7117. Dixon, RAF, et al. 1987. Ligand binding to the...
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Signal Transduction

Carl-Henrik Heldin, Mary Purton - 1996 - 404 páginas
...muscatinic receptor. Annu. Ree. Neurosri., 10. 195-236. 14 De Lean A., StadeL JM and Letkowitz, RJ (1980l A ternary complex model explains the agonist-specific...binding properties of the adenylate cyclase-coupled p-adrenergic receptor. J. Biol Chem., 255, 7108-17. 15 Samama, P., Cotecchia, S., Costa, T. and Leflcowitz,...
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alpha2Adrenergic Receptors

Lewis L. Lanier - 1997 - 234 páginas
...function. Proc. Nail Acad. Sci. USA. 87. 2896-2900. De Lean. A.. Stadel. JM and Lefkowitz, RJ (1980). A ternary complex model explains the agonist-specific...binding properties of the adenylate cyclase-coupled p-adrenergic receptor. J. Biol Chem.. 255. 7 1 08-7 1 1 7. Hess. P.. Lansman. JB and Tsien. RW ( 1984)....
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Muscarinic Receptor Subtypes in Smooth Muscle

Richard M. Eglen - 1997 - 212 páginas
...sitedirected mutagenesis. Eur. ]. Pharmacol. 289, 429, 1995. 44. DeLean, A., Stadel, JM, and Lefkowitz, RJ A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase coupled p-adrenergic receptor. /. Biol. Chem. 255, 7108, 1980. 45. Birdsall, NJM, Burgen, ASV,...
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Dopamine Receptor Subtypes: From Basic Science to Clinical Application

Peter Jenner, R. Demirdamar - 1998 - 200 páginas
...of exploratinn? A critical review. Psychopharmacology, iBerl > 106 11992) 1,13. [22] A. DeLean et al A ternary complex model explains the agonist,specific...binding properties of the adenylate cyclase,coupled ft,adrenergic receptor. J. Biol Chem 255119g0)710g.7117. [23] T. Costa et ai Drug efficacy at guanine...
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Receptor Binding Techniques

Mary Keen - 1999 - 288 páginas
...protein subunits. Mol. Pharmacol. 43, 245-256. 38. De Lean, A., Stadel, JM, and Lefkowitz, RJ (1980) A ternary complex model explains the agonist-specific...cyclase-coupled beta-adrenergic receptor. J. Biol. Chem. 255, 7108-71 17. 39. Sim, LJ, Selley, DE, Xiao, R., and Childers, SR (1996) Differences in G-protein...
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Quantitative Molecular Pharmacology and Informatics in Drug Discovery

Michael Lutz, Terry Kenakin - 2000 - 438 páginas
...«iB-adrenergic receptor. Binchem Soc Trans 23: 121-125. De Lean A, Kilpatrick BF and Carón M (1982) A ternary complex model explains the agonist-specific...binding properties of the adenylate cyclase-coupled /J-adrencrgic receptor. J Biol Chem 255: 7108-7117. Freissmuth M, Selzer E and Schutz W ( 1 99 1 )...
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